Design and synthesis of human immunodeficiency virus entry inhibitors: Sulfonamide as an isostere for the α-ketoamide group

Rong Jian Lu, John A. Tucker, Tatiana Zinevitch, Olga Kirichenko, Vitalii Konoplev, Svetlana Kuznetsova, Sergey Sviridov, Jason Pickens, Sagun Tandel, Enugurthi Brahmachary, Yang Yang, Jian Wang, Stephanie Freel, Shelly Fisher, Alana Sullivan, Jiying Zhou, Sherry Stanfield-Oakley, Michael Greenberg, Dani Bolognesi, Brian BrayBarney Koszalka, Peter Jeffs, Alisher Khasanov, You An Ma, Cynthia Jeffries, Changhui Liu, Tatiana Proskurina, Tong Zhu, Alexander Chucholowski, Rongshi Li, Connie Sexton

Research output: Contribution to journalArticle

53 Scopus citations
Original languageEnglish (US)
Pages (from-to)6535-6544
Number of pages10
JournalJournal of Medicinal Chemistry
Volume50
Issue number26
DOIs
Publication statusPublished - Dec 27 2007

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ASJC Scopus subject areas

  • Molecular Medicine
  • Drug Discovery

Cite this

Lu, R. J., Tucker, J. A., Zinevitch, T., Kirichenko, O., Konoplev, V., Kuznetsova, S., ... Sexton, C. (2007). Design and synthesis of human immunodeficiency virus entry inhibitors: Sulfonamide as an isostere for the α-ketoamide group. Journal of Medicinal Chemistry, 50(26), 6535-6544. https://doi.org/10.1021/jm070650e